Molecule Details
InChIKeyCFSZFZQNXIYCLF-IBGZPJMESA-N
Canonical SMILESC=C1C[C@@H](c2nc3cccc(C)c3[nH]2)N(C(=O)c2nc(C)sc2-c2ccc(F)c(Br)c2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.41
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
O43614 HCRTR2 Homo sapiens Human PF00001 PF03827 9.0 IC50 ChEMBL;BindingDB
O43613 HCRTR1 Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB