Molecule Details
InChIKeyCEWKJGUDXOKCAF-UHFFFAOYSA-N
Compound Name2-(4-fluoro-2-methylphenoxy)-N-(2-methyl-6-oxo-1H-pyridin-4-yl)-5-(trifluoromethyl)benzamide
Canonical SMILESCc1cc(NC(=O)c2cc(C(F)(F)F)ccc2Oc2ccc(F)cc2C)cc(=O)[nH]1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.95
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UQD0 SCN8A Homo sapiens Human PF00520 PF24609 PF06512 PF11933 7.0 IC50 ChEMBL;BindingDB
Q9Y5Y9 SCN10A Homo sapiens Human PF00520 PF24609 PF06512 7.0 IC50 ChEMBL;BindingDB