Molecule Details
InChIKeyCEVDMQKZKKCGLK-HMILPKGGSA-N
Compound Namemethyl (2R,15R)-2-[(1-aminoisoquinolin-6-yl)amino]-4,15,17-trimethyl-3,12-dioxo-13-oxa-4,11-diazatricyclo[14.2.2.16,10]henicosa-1(18),6,8,10(21),16,19-hexaene-7-carboxylate
Canonical SMILESCOC(=O)c1ccc2cc1CN(C)C(=O)[C@H](Nc1ccc3c(N)nccc3c1)c1ccc(c(C)c1)[C@@H](C)COC(=O)N2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.57
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08709 F7 Homo sapiens Human PF00008 PF14670 PF00594 PF00089 8.1 Ki ChEMBL;BindingDB
P13726 F3 Homo sapiens Human PF09294 PF01108 8.1 Ki ChEMBL
P06870 KLK1 Homo sapiens Human PF00089 6.6 Ki ChEMBL;BindingDB