Molecule Details
InChIKeyCETJSTBZOJQTPJ-UHFFFAOYSA-N
Compound Name8-(2-Fluorophenyl)-7-hydroxy-4-(3-imidazol-1-ylphenyl)-1,3-dihydro-1,5-benzodiazepin-2-one
Canonical SMILESO=C1CC(c2cccc(-n3ccnc3)c2)=Nc2cc(O)c(-c3ccccc3F)cc2N1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.28
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P08684 CYP3A4 Homo sapiens Human PF00067 9.0 IC50 ChEMBL;BindingDB
Q14416 GRM2 Homo sapiens Human PF00003 PF01094 PF07562 7.6 IC50 BindingDB