Molecule Details
InChIKeyCEJFYMKXALJHTD-UHFFFAOYSA-N
Compound Name3-(2-(4-(2-Methyl-2H-tetrazol-5-yl)phenylamino)pyrimidin-4-yl)-5-morpholinobenzonitrile
Canonical SMILESCn1nnc(-c2ccc(Nc3nccc(-c4cc(C#N)cc(N5CCOCC5)c4)n3)cc2)n1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.1
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45983 MAPK8 Homo sapiens Human PF00069 7.3 IC50 ChEMBL;BindingDB
P53779 MAPK10 Homo sapiens Human PF00069 6.8 IC50 ChEMBL;BindingDB