Molecule Details
InChIKeyCEFDHULRYUTNDO-UHFFFAOYSA-N
Compound NameN-(4-(methylsulfonyl)benzyl)-4-amino-6-ethoxy-5-ethynylpicolinamide
Canonical SMILESC#Cc1c(N)cc(C(=O)NCc2ccc([S@SP2](C)(=O)=O)cc2)nc1OCC
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL6.49
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P45984 MAPK9 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB
P45983 MAPK8 Homo sapiens Human PF00069 6.5 IC50 ChEMBL;BindingDB