Molecule Details
InChIKeyCEEARFKAZMLMSC-NOCPHRDISA-N
Compound NameSuc-Asp-Glu-Phe(2-Me)-Gly(tBu)-Leu-D-Nle-CONH2
Canonical SMILESCCCC[C@@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1ccccc1C)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC(=O)O)NC(=O)CCC(=O)O)C(C)(C)C)C(=O)C(N)=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.48
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q99895 CTRC Homo sapiens Human PF00089 6.5 IC50 ChEMBL;BindingDB
A3EZI9 NS3 Hepacivirus hominis Pathogen PF07652 PF22027 PF02907 8.0 IC50 ChEMBL;BindingDB
D2K2A8 NS4A Hepacivirus hominis Pathogen PF01006 8.0 IC50 ChEMBL