Molecule Details
InChIKeyCEANXNAMUUCBQK-UHFFFAOYSA-N
Canonical SMILESCn1cc(-c2ccc3cnc(Nc4ccc(-n5cnc(N6CCOCC6)n5)cc4)nc3c2-c2ccccc2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P53779 MAPK10 Homo sapiens Human PF00069 8.0 IC50 ChEMBL;BindingDB
P05412 JUN Homo sapiens Human PF00170 PF03957 7.4 IC50 ChEMBL;BindingDB