Molecule Details
InChIKeyCEABWOSUDRMZCJ-UHFFFAOYSA-N
Compound NameN-(7-(N-ethylacetamido)-4-methoxybenzo[d]thiazol-2-yl)-1-(3-(trifluoromethyl)benzyl)-1H-pyrazole-4-carboxamide
Canonical SMILESCCN(C(C)=O)c1ccc(OC)c2nc(NC(=O)c3cnn(Cc4cccc(C(F)(F)F)c4)c3)sc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29274 ADORA2A Homo sapiens Human PF00001 8.5 Ki ChEMBL;BindingDB
P29275 ADORA2B Homo sapiens Human PF00001 8.3 IC50 ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 8.2 Ki ChEMBL;BindingDB