Molecule Details
InChIKeyCDXIZXQBISVZMK-VWLOTQADSA-N
Compound Name4-[5-({(3-Amino-propyl)-[1-(3-chloro-benzyl)-2-oxo-pyrrolidin-3-yl]-amino}-methyl)-imidazol-1-ylmethyl]-benzonitrile
Canonical SMILESN#Cc1ccc(Cn2cncc2CN(CCCN)[C@H]2CCN(Cc3cccc(Cl)c3)C2=O)cc1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.79
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.1 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.5 IC50 ChEMBL;BindingDB