Molecule Details
InChIKeyCDWUOIQIYZWIIH-UHFFFAOYSA-N
Compound Name1-Cyclopropyl-6-fluoro-7-[4-[1-[4-[(5-methyl-1,2-oxazol-3-yl)sulfamoyl]anilino]-1-oxopropan-2-yl]piperazin-1-yl]-4-oxoquinoline-3-carboxylic acid
Canonical SMILESCc1cc(NS(=O)(=O)c2ccc(NC(=O)C(C)N3CCN(c4cc5c(cc4F)c(=O)c(C(=O)O)cn5C4CC4)CC3)cc2)no1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL6.41
SourceChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P0C1S7 parE Staphylococcus aureus Pathogen PF00204 PF00986 PF02518 PF01751 6.4 IC50 ChEMBL
P0C1U9 parC Staphylococcus aureus Pathogen PF03989 PF00521 6.4 IC50 ChEMBL