Molecule Details
InChIKeyCDUXPGVKEOGWKB-UHFFFAOYSA-N
Compound Name1,4-diazabicyclo[3.2.2]nonan-4-yl-[3-(4-fluorophenyl)-5,7-dihydro-4H-pyrano[4,3-d]pyrazol-1-yl]methanone
Canonical SMILESO=C(N1CCN2CCC1CC2)n1nc(-c2ccc(F)cc2)c2c1COCC2
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL7.06
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q16739 UGCG Homo sapiens Human PF13506 7.5 IC50 ChEMBL;BindingDB
P46098 HTR3A Homo sapiens Human PF02931 PF02932 6.7 IC50 ChEMBL;BindingDB