Molecule Details
InChIKeyCDNFAKVJGFHDDB-UHFFFAOYSA-N
Compound Name1-(5-{3,5-Bis[5-(3-phenylpyridin-1-ium-1-yl)pentyl]phenyl}pentyl)-3-phenylpyridin-1-ium tribromide
Canonical SMILESc1ccc(-c2ccc[n+](CCCCCc3cc(CCCCC[n+]4cccc(-c5ccccc5)c4)cc(CCCCC[n+]4cccc(-c5ccccc5)c4)c3)c2)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.85
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9GZZ6 CHRNA10 Homo sapiens Human PF02931 PF02932 9.2 IC50 ChEMBL;BindingDB
Q9UGM1 CHRNA9 Homo sapiens Human PF02931 PF02932 9.2 IC50 ChEMBL
P36544 CHRNA7 Homo sapiens Human PF02931 PF02932 8.1 IC50 ChEMBL;BindingDB