Molecule Details
InChIKeyCCOWQXCHSULBCV-UHFFFAOYSA-N
Compound NameUS11066396, Example 420
Canonical SMILESCOCc1cc(=O)n(Cc2ccc(-c3noc(C(F)(F)F)n3)cn2)c2ccccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.13
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 8.4 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 7.0 IC50 ChEMBL;BindingDB
Q9BY41 HDAC8 Homo sapiens Human PF00850 6.0 IC50 ChEMBL;BindingDB