Molecule Details
InChIKeyCBZNDVANLGVAAJ-UHFFFAOYSA-N
Compound Name8-(5-Fluoroazepan-4-yl)oxy-2-([1,2,4]triazolo[4,3-a]pyridin-3-yl)quinoline
Canonical SMILESFC1CCNCCC1Oc1cccc2ccc(-c3nnc4ccccn34)nc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.96
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 9.0 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.9 IC50 ChEMBL;BindingDB