Molecule Details
InChIKeyCBZLQUNISFBVLM-UHFFFAOYSA-N
Compound Name4-[2-[5,7,12,14-Tetraoxo-13-(2-sulfamoylethyl)-6,13-diazatetracyclo[6.6.2.04,16.011,15]hexadeca-1(15),2,4(16),8,10-pentaen-6-yl]ethyl]benzenesulfonamide
Canonical SMILESNS(=O)(=O)CCN1C(=O)c2ccc3c4c(ccc(c24)C1=O)C(=O)N(CCc1ccc(S(N)(=O)=O)cc1)C3=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O43570 CA12 Homo sapiens Human PF00194 7.7 Ki ChEMBL;BindingDB
Q16790 CA9 Homo sapiens Human PF00194 7.6 Ki ChEMBL;BindingDB
P00918 CA2 Homo sapiens Human PF00194 6.8 Ki ChEMBL;BindingDB