Molecule Details
InChIKeyCBPBGAAUJILPTQ-UHFFFAOYSA-N
Compound NameN-ethyl-4-methyl-1-pyridin-2-yl-[1,2,4]triazolo[4,3-a]quinoxaline-8-carboxamide
Canonical SMILESCCNC(=O)c1ccc2nc(C)c3nnc(-c4ccccn4)n3c2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.14
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9Y233 PDE10A Homo sapiens Human PF01590 PF00233 7.7 IC50 ChEMBL;BindingDB
O00408 PDE2A Homo sapiens Human PF01590 PF00233 6.6 IC50 ChEMBL;BindingDB