Molecule Details
InChIKeyCBGMGQVEMRTNGL-VQTJNVASSA-N
Compound Nametrans-(1R,2R)-N-[4-(1-propylpyrazol-4-yl)sulfonylphenyl]-2-pyridin-3-ylcyclopropane-1-carboxamide
Canonical SMILESCCCn1cc(S(=O)(=O)c2ccc(NC(=O)[C@@H]3C[C@H]3c3cccnc3)cc2)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.92
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43490 NAMPT Homo sapiens Human PF18127 PF04095 8.1 IC50 ChEMBL;BindingDB
P08684 CYP3A4 Homo sapiens Human PF00067 6.6 IC50 ChEMBL
P11712 CYP2C9 Homo sapiens Human PF00067 6.0 IC50 ChEMBL;BindingDB