Molecule Details
InChIKeyCBGFEMSXMIJQKG-UHFFFAOYSA-N
Compound Name6-but-3-enyl-4-[3-methyl-7-(morpholine-4-carbonyl)benzimidazol-5-yl]-1H-pyrrolo[2,3-c]pyridin-7-one
Canonical SMILESC=CCCn1cc(-c2cc(C(=O)N3CCOCC3)c3ncn(C)c3c2)c2cc[nH]c2c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.29
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9BXF3 CECR2 Homo sapiens Human PF00439 8.0 IC50 ChEMBL;BindingDB
P21675 TAF1 Homo sapiens Human PF00439 PF12157 PF09247 PF15288 7.8 IC50 ChEMBL;BindingDB
Q9H8M2 BRD9 Homo sapiens Human PF00439 PF12024 6.1 IC50 ChEMBL;BindingDB