Molecule Details
InChIKeyCBEJYUZNCXVSSY-UHFFFAOYSA-N
Compound Name6-[(2-Methoxy-5-methylphenylamino)methyl]-2,4-diamino-5-methylpyrido[2,3-d]pyrimidine
Canonical SMILESCOc1ccc(C)cc1NCc1cnc2nc(N)nc(N)c2c1C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.8
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P00374 DHFR Homo sapiens Human PF00186 6.5 IC50 ChEMBL;BindingDB
O30463 folA Mycobacterium avium Pathogen PF00186 9.1 IC50 ChEMBL
Q07422 Toxoplasma gondii Pathogen PF00186 PF00303 7.8 IC50 ChEMBL;BindingDB