Molecule Details
InChIKeyCAZNIOSROXHNKZ-UHFFFAOYSA-N
Compound Name8-(4-Piperidinylmethoxy)-2-(1,2,4-triazolo[4,3-a]pyridin-3-yl)quinoline
Canonical SMILESc1cc(OCC2CCNCC2)c2nc(-c3nnc4ccccn34)ccc2c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.47
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11309 PIM1 Homo sapiens Human PF00069 8.7 IC50 ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 6.2 IC50 ChEMBL;BindingDB