Molecule Details
InChIKeyCAVUPJAIIXVCRJ-HXWGMKPQSA-N
Compound Name2-[13-(4-Amino-butyl)-7,22-dibenzyl-10-(1-hydroxy-ethyl)-16,19-bis-(1H-indol-3-ylmethyl)-6,9,12,15,18,21,24-heptaoxo-1,2-dithia-5,8,11,14,17,20,23-heptaaza-cyclopentacos-5-yl]-acetamide
Canonical SMILESC[C@@H](O)[C@@H]1NC(=O)[C@@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)CSSCCN(CC(N)=O)C(=O)[C@@H](Cc2ccccc2)NC1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.08
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35346 SSTR5 Homo sapiens Human PF00001 8.9 IC50 ChEMBL;BindingDB
P32745 SSTR3 Homo sapiens Human PF00001 7.8 IC50 ChEMBL;BindingDB
P30874 SSTR2 Homo sapiens Human PF00001 7.5 IC50 ChEMBL;BindingDB