Molecule Details
InChIKeyCAIDLKSVZKWPJK-LSDHHAIUSA-N
Compound Name2-[[(1R,2S)-2-aminocyclohexyl]amino]-4-(4-methylanilino)pyrimidine-5-carboxamide
Canonical SMILESCc1ccc(Nc2nc(N[C@@H]3CCCC[C@@H]3N)ncc2C(N)=O)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.4
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P43405 SYK Homo sapiens Human PF07714 PF00017 8.0 IC50 ChEMBL;BindingDB
P27361 MAPK3 Homo sapiens Human PF00069 7.1 IC50 ChEMBL
P28482 MAPK1 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB