Molecule Details
InChIKeyCAGHIASAHLPQMS-UHFFFAOYSA-N
Compound NameN-cyclopropyl-4-pyrazolo(1,5-b)pyridazin-3-ylpyrimidin-2-amine
Canonical SMILESc1cnn2ncc(-c3ccnc(NC4CC4)n3)c2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.01
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
DrugBank Annotations
DrugBank ID DB07164
Drug NameN-cyclopropyl-4-pyrazolo[1,5-b]pyridazin-3-ylpyrimidin-2-amine
CAS Numbernan
Groups experimental
ATC Codes nan
Descriptionnan

Cross-references: BindingDB: 50293162 CHEMBL525194 ChemSpider: 5293903 PDB: 5BP PubChem:6918710 PubChem:99443635 ZINC: ZINC000020149019
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P11802 CDK4 Homo sapiens Human PF00069 7.1 IC50 ChEMBL;BindingDB
P24941 CDK2 Homo sapiens Human PF00069 6.9 pIC50 TTD_MultiTarget
DrugBank Target Actions (2)
Target Gene Target Name Action Type
P20248 CCNA2 Cyclin-A2 binder targets
P24941 CDK2 Cyclin-dependent kinase 2 binder targets