Molecule Details
InChIKeyBYPUTAKAOUIYHF-ZDUSSCGKSA-N
Compound NameN-((3S)-1-(6-(aminomethyl)-5-(2,4-dichlorophenyl)-7-methylimidazo[1,2-a]pyrimidine-2-carbonyl)pyrrolidin-3-yl)methanesulfonamide
Canonical SMILESCc1nc2nc(C(=O)N3CC[C@H](NS(C)(=O)=O)C3)cn2c(-c2ccc(Cl)cc2Cl)c1CN
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.02
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P27487 DPP4 Homo sapiens Human PF00930 PF00326 9.7 Ki ChEMBL;BindingDB
Q6V1X1 DPP8 Homo sapiens Human PF19520 PF00930 PF00326 8.7 Ki ChEMBL;BindingDB
Q86TI2 DPP9 Homo sapiens Human PF19520 PF00930 PF00326 8.7 Ki ChEMBL;BindingDB