Molecule Details
InChIKeyBXZWRAYRDLNDSN-UHFFFAOYSA-N
Compound Name6-(4-(4-(2-isopropoxyphenyl)piperazin-1-yl)cyclohexyl)-6H-pyrrolo[3,4-b]pyridine-5,7-dione
Canonical SMILESCC(C)Oc1ccccc1N1CCN(C2CCC(N3C(=O)c4cccnc4C3=O)CC2)CC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.42
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P35348 ADRA1A Homo sapiens Human PF00001 9.1 Ki ChEMBL;BindingDB
P25100 ADRA1D Homo sapiens Human PF00001 8.8 Ki ChEMBL;BindingDB
P35368 ADRA1B Homo sapiens Human PF00001 7.3 Ki ChEMBL;BindingDB