Molecule Details
InChIKeyBXMUAQLRVCWTKG-UHFFFAOYSA-N
Compound Name3-[5-Ethyl-5-(2-furyl)-2-oxo-1,2,3,5-tetrahydro-4,1-benzoxazepin-7-yl]-5-fluorobenzonitrile
Canonical SMILESCCC1(c2ccco2)OCC(=O)Nc2ccc(-c3cc(F)cc(C#N)c3)cc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.94
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P06401 PGR Homo sapiens Human PF00104 PF02161 PF00105 7.9 IC50 ChEMBL;BindingDB
P04150 NR3C1 Homo sapiens Human PF02155 PF00104 PF00105 6.7 IC50 ChEMBL;BindingDB
P10275 AR Homo sapiens Human PF02166 PF00104 PF00105 6.2 IC50 ChEMBL;BindingDB