Molecule Details
InChIKeyBWXIPDFABPPPPW-CXAGYDPISA-N
Canonical SMILESCCc1cccc(-c2c(-c3ccc4nn(C)cc4c3)nsc2NC(=O)[C@@H]2C[C@H]2C)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.28
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P41594 GRM5 Homo sapiens Human PF00003 PF01094 PF10606 PF07562 8.0 IC50 ChEMBL;BindingDB
Q13255 GRM1 Homo sapiens Human PF00003 PF01094 PF10606 PF07562 6.5 IC50 ChEMBL;BindingDB