Molecule Details
InChIKeyBWLYGOVEEHWYDU-UHFFFAOYSA-N
Compound Name1-(Cyclopropyl)methyl-5-isopropyl-6-(3,5-dimethylphenoxy)-2,4-pyrimidinedione
Canonical SMILESCc1cc(C)cc(Oc2c(C(C)C)c(=O)[nH]c(=O)n2CC2CC2)c1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.73
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9WKE8 reverse transcriptase Human immunodeficiency virus type 1 Pathogen PF00078 7.9 IC50 BindingDB
Q72547 pol Human immunodeficiency virus type 1 Pathogen PF00075 PF00078 PF06815 PF06817 7.5 IC50 ChEMBL