Molecule Details
InChIKeyBWIBKWVUAHMKER-UHFFFAOYSA-N
Compound Name(-)-2-Chloro-4b-methyl-4b,5,6,10-tetrahydrophenanthrene-7-carboxylic acid
Canonical SMILESCC12CCC(C(=O)O)=CC1=CCc1cc(Cl)ccc12
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL6.59
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P18505 GABRB1 Homo sapiens Human PF02931 PF02932 6.6 pIC50 TTD_MultiTarget
P31639 SLC5A2 Homo sapiens Human PF00474 6.6 pIC50 TTD_MultiTarget
P31213 SRD5A2 Homo sapiens Human PF02544 6.6 Ki ChEMBL