Molecule Details
InChIKeyBVWYBVKUPUODDY-QOBPCVTDSA-N
Compound Name1-(2-((R)-4-(6-fluoronaphthalen-1-yl)-2-methylpiperazin-1-yl)ethyl)-3,4-dihydro-1H-isochromene-6-carboxamide
Canonical SMILESC[C@@H]1CN(c2cccc3cc(F)ccc23)CCN1CCC1OCCc2cc(C(N)=O)ccc21
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.63
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P31645 SLC6A4 Homo sapiens Human PF03491 PF00209 9.1 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 7.2 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 6.5 Ki ChEMBL;BindingDB