Molecule Details
InChIKeyBVWSIHNUHWGLEX-UHFFFAOYSA-N
Compound Name8-(1-((3-phenyl-1,2,4-oxadiazol-5-yl)methyl)-1H-pyrazol-4-yl)-1,3-dipropyl-1H-purine-2,6(3H,7H)-dione
Canonical SMILESCCCn1c(=O)c2nc(-c3cnn(Cc4nc(-c5ccccc5)no4)c3)[nH]c2n(CCC)c1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.25
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P29275 ADORA2B Homo sapiens Human PF00001 9.0 Ki ChEMBL;BindingDB
P30542 ADORA1 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P0DMS8 ADORA3 Homo sapiens Human PF00001 6.3 Ki ChEMBL;BindingDB