Molecule Details
InChIKeyBVHVEJVRGYHQTC-XFTNXAEASA-N
Compound Name(2S)-2-[[(2R)-2-[(7S)-7-acetamido-6-oxo-7,8-dihydro-4H-triazolo[1,5-a][1,4]diazepin-5-yl]-3-phenylpropanoyl]amino]-N-[(2S)-1-amino-3-(1H-indol-3-yl)-1-oxopropan-2-yl]-5-(diaminomethylideneamino)pentanamide
Canonical SMILESCC(=O)N[C@H]1Cn2nncc2CN([C@H](Cc2ccccc2)C(=O)N[C@@H](CCCNC(=N)N)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(N)=O)C1=O
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.52
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P33032 MC5R Homo sapiens Human PF00001 6.9 IC50 ChEMBL;BindingDB
P32245 MC4R Homo sapiens Human PF00001 6.7 IC50 ChEMBL;BindingDB
P41968 MC3R Homo sapiens Human PF00001 6.0 IC50 ChEMBL;BindingDB