Molecule Details
InChIKeyBVCQRIMNJALALQ-CNNODRBYSA-N
Compound Name(S)-4-Carbamoyl-2-({(S)-2-[(S)-2-(2-3H-imidazol-4-yl-acetylamino)-3,3-dimethyl-butyryl]-1,2,3,4-tetrahydro-isoquinoline-3-carbonyl}-amino)-butyric acid
Canonical SMILESCC(C)(C)[C@H](NC(=O)Cc1c[nH]cn1)C(=O)N1Cc2ccccc2C[C@H]1C(=O)N[C@@H](CCC(N)=O)C(=O)O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Cross-Family
Avg pChEMBL7.55
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 7.5 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 7.5 IC50 ChEMBL;BindingDB
P53609 PGGT1B Homo sapiens Human PF00432 7.5 IC50 ChEMBL