Molecule Details
InChIKeyBTJDQFBAKDDPOT-UXHICEINSA-N
Compound Name(3R,5S)-N-benzyl-1-[(6-methoxy-3-pyridinyl)methyl]-3,5-dimethyl-3,5-dihydro-2H-1,4-benzodiazepine-4-carboxamide
Canonical SMILESCOc1ccc(CN2C[C@@H](C)N(C(=O)NCc3ccccc3)[C@@H](C)c3ccccc32)cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.61
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9P0X4 CACNA1I Homo sapiens Human PF00520 8.0 IC50 ChEMBL;BindingDB
O95180 CACNA1H Homo sapiens Human PF00520 7.5 IC50 ChEMBL;BindingDB
O43497 CACNA1G Homo sapiens Human PF00520 7.3 IC50 ChEMBL;BindingDB