Molecule Details
InChIKeyBSUWUKYJNUNGOM-CAMINTRRSA-N
Canonical SMILESCCC(CC)C(NC(=O)CN1C[C@H](c2ccc3c(c2)OCO3)[C@@H](C(=O)O)[C@@H]1c1ccc(OC)cc1)c1ccccc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL8.78
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P24530 EDNRB Homo sapiens Human PF00001 9.0 IC50 ChEMBL;BindingDB
P25101 EDNRA Homo sapiens Human PF00001 8.6 IC50 ChEMBL;BindingDB