Molecule Details
InChIKeyBSFNGHCTZDCQBF-ZUICHYAESA-N
Compound Name(3E)-5-(5-{[(2S)-2-amino-3-(1H-indol-3-yl)propyl]oxy}pyridin-3-yl)-3-(furan-2-ylmethylidene)-1,3-dihydro-2H-indol-2-one
Canonical SMILESN[C@H](COc1cncc(-c2ccc3c(c2)/C(=C\c2ccco2)C(=O)N3)c1)Cc1c[nH]c2ccccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.29
SourceBindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q9NYY3 PLK2 Homo sapiens Human PF00069 PF00659 6.8 Ki BindingDB
Q9H4B4 PLK3 Homo sapiens Human PF00069 PF00659 6.0 Ki BindingDB
O00444 PLK4 Homo sapiens Human PF00069 PF18190 PF18409 6.0 Ki BindingDB