Molecule Details
InChIKeyBSFBSBUVPRPQFW-UHFFFAOYSA-N
Compound Name6-[Amino-(4-chloro-phenyl)-(3-methyl-3H-imidazol-4-yl)-methyl]-4-(3-chloro-phenyl)-1H-quinolin-2-one
Canonical SMILESCn1cncc1C(N)(c1ccc(Cl)cc1)c1ccc2nc(O)cc(-c3cccc(Cl)c3)c2c1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)2
Pfam Stratification Cross-Family
Avg pChEMBL8.46
SourceChEMBL;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P49354 FNTA Homo sapiens Human PF01239 8.5 pIC50 TTD_MultiTarget
P49356 FNTB Homo sapiens Human PF00432 8.5 IC50 ChEMBL