Molecule Details
InChIKeyBSACLFCWNMRHBP-DRFRAUJUSA-N
Compound Name(1R,3R,6R,7S,8R,10S,11S,14R,15S,20S)-8-hydroxy-7-[(1S)-1-[(2-methoxyphenyl)methyl-methylamino]ethyl]-6,10,15-trimethyl-18-propan-2-yl-17-thia-19-azahexacyclo[12.8.0.01,3.03,11.06,10.015,20]docos-18-en-4-one
Canonical SMILESCOc1ccccc1CN(C)[C@@H](C)[C@H]1[C@H](O)C[C@@]2(C)[C@@H]3CC[C@H]4[C@]5(C)CSC(C(C)C)=N[C@H]5CC[C@@]45C[C@@]35C(=O)C[C@]12C
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)2
Pfam Stratification Homologous
Avg pChEMBL7.35
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (2)
Target Gene Organism Category Pfam pChEMBL Type Source
P22303 ACHE Homo sapiens Human PF08674 PF00135 8.2 IC50 ChEMBL;BindingDB
P06276 BCHE Homo sapiens Human PF08674 PF00135 6.5 IC50 ChEMBL;BindingDB