Molecule Details
InChIKeyBQVZFNYKORVNKX-CQSZACIVSA-N
Compound Name(3R)-1-[6-[6-(1,3-thiazol-5-yl)pyrazolo[4,3-c]pyridin-1-yl]-2-pyridinyl]piperidin-3-amine
Canonical SMILESN[C@@H]1CCCN(c2cccc(-n3ncc4cnc(-c5cncs5)cc43)n2)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL9.03
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q86V86 PIM3 Homo sapiens Human PF00069 9.4 Ki ChEMBL;BindingDB
P11309 PIM1 Homo sapiens Human PF00069 9.3 Ki ChEMBL;BindingDB
Q9P1W9 PIM2 Homo sapiens Human PF00069 8.3 Ki ChEMBL;BindingDB