Molecule Details
InChIKeyBQLIAGXOCFHIGO-UHFFFAOYSA-N
Compound Name4-{3-[(4,5,6,7-Tetrahydro-pyrazolo[1,5-a]pyrazine-3-carbonyl)-amino]-benzylamino}-quinazoline-8-carboxylic acid amide
Canonical SMILESNC(=O)c1cccc2c(NCc3cccc(NC(=O)c4cnn5c4CNCC5)c3)ncnc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.87
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
Q96GD4 AURKB Homo sapiens Human PF00069 8.8 IC50 ChEMBL;BindingDB
O14965 AURKA Homo sapiens Human PF00069 8.1 IC50 ChEMBL;BindingDB
P23443 RPS6KB1 Homo sapiens Human PF00069 PF00433 6.8 IC50 ChEMBL;BindingDB