Molecule Details
InChIKeyBOXRBFJLKOMZNE-UHFFFAOYSA-N
Compound Name7-fluoro-N,N-dimethyl-3-((2-(tetrahydro-2H-pyran-4-yl)ethylamino)methyl)-3,4-dihydro-2H-benzo[b][1,4]dioxepin-3-amine
Canonical SMILESCN(C)C1(CNCCC2CCOCC2)COc2ccc(F)cc2OC1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.04
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P20309 CHRM3 Homo sapiens Human PF00001 8.4 Ki ChEMBL;BindingDB
P08172 CHRM2 Homo sapiens Human PF00001 8.3 Ki ChEMBL;BindingDB
P11229 CHRM1 Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB