Molecule Details
InChIKeyBOWWSMXUIIXBOU-ZHACJKMWSA-N
Compound NameN-(6-(pyrrolidin-1-yl)-3-styryl-1H-indazol-5-yl)-2-(thiophen-2-yl)acetamide
Canonical SMILESO=C(Cc1cccs1)Nc1cc2c(/C=C/c3ccccc3)n[nH]c2cc1N1CCCC1
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.01
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
O14965 AURKA Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB
O75716 STK16 Homo sapiens Human PF00069 7.0 pIC50 TTD_MultiTarget
Q96GD4 AURKB Homo sapiens Human PF00069 7.0 IC50 ChEMBL;BindingDB