Molecule Details
InChIKeyBNMIOTKQNUSAEJ-UHFFFAOYSA-N
Compound Name2-[3-(2-Amino-ethyl)-1H-indol-5-yloxy]-1-(4-{2-[3-(2-amino-ethyl)-1H-indol-5-yloxy]-acetyl}-piperazin-1-yl)-ethanone
Canonical SMILESNCCc1c[nH]c2ccc(OCC(=O)N3CCN(C(=O)COc4ccc5[nH]cc(CCN)c5c4)CC3)cc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.84
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P28222 HTR1B Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 9.4 Ki ChEMBL;BindingDB
P08908 HTR1A Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB