Molecule Details
InChIKeyBMZBCRXOQLRHKH-UHFFFAOYSA-N
Compound NameUS9670193, 11 N-((6-methylpyridin-2-yl)methyl)-5-(5-(trifluoromethyl)-1,2,4-oxadiazol-3-yl)pyrimidin-2-amine
Canonical SMILESCc1cccc(CNc2ncc(-c3noc(C(F)(F)F)n3)cn2)n1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.39
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P56524 HDAC4 Homo sapiens Human PF12203 PF00850 6.6 IC50 ChEMBL;BindingDB
Q13547 HDAC1 Homo sapiens Human PF00850 6.3 IC50 ChEMBL;BindingDB
Q9UBN7 HDAC6 Homo sapiens Human PF00850 PF02148 6.3 IC50 ChEMBL;BindingDB