Molecule Details
InChIKeyBMTFZBSAMOYHLW-UHFFFAOYSA-N
Compound Name6-(3-sulfamoyl-2-(2H-tetrazol-5-yl)phenyl)isoquinoline-1-carboxamide
Canonical SMILESNC(=O)c1nccc2cc(-c3cccc(S(N)(=O)=O)c3-c3nn[nH]n3)ccc12
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.25
SourceBindingDB;ChEMBL
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
C7C422 blaNDM-1 Klebsiella pneumoniae Pathogen PF00753 9.5 IC50 ChEMBL;BindingDB
Q5GN09 vim-1 Klebsiella pneumoniae Pathogen PF00753 7.9 IC50 BindingDB
P52699 Serratia marcescens Pathogen PF00753 7.4 IC50 BindingDB