Molecule Details
InChIKeyBMLRTLPESFVXBM-UHFFFAOYSA-N
Compound NameN-[4-(4-pyridin-2-ylpiperazin-1-yl)butyl]isoquinoline-3-carboxamide
Canonical SMILESO=C(NCCCCN1CCN(c2ccccn2)CC1)c1cc2ccccc2cn1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.09
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 7.8 Ki ChEMBL;BindingDB
P35462 DRD3 Homo sapiens Human PF00001 7.4 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.1 Ki ChEMBL;BindingDB