Molecule Details
InChIKeyBMCUOUFSLYKUKP-UHFFFAOYSA-N
Compound Name1-[1-(4-Cyanophenyl)-5-ethylpyrazol4-ylcarbonyl]-2,3-dihydro-8-(piperazin-1-yl)pyrrolo[3,2-g]isoquinoline
Canonical SMILESCCc1c(C(=O)N2CCc3cc4ccnc(N5CCNCC5)c4cc32)cnn1-c1ccc(C#N)cc1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL8.7
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 8.9 Ki ChEMBL;BindingDB
P28221 HTR1D Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB
P28222 HTR1B Homo sapiens Human PF00001 8.6 Ki ChEMBL;BindingDB