Molecule Details
InChIKeyBMCMQADGLVGIMX-UHFFFAOYSA-N
Compound NameN-[1-[4'-(Trifluoromethyl)-4-biphenylyloxymethyl]-2-(2,5-dioxo-4,4-dimethylimidazolidine-1-yl)ethyl]formhydroxamic acid
Canonical SMILESCC1(C)NC(=O)N(CC(COc2ccc(-c3ccc(C(F)(F)F)cc3)cc2)N(O)C=O)C1=O
Clinical Status Clinical Multi-Target
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL7.16
SourceChEMBL;BindingDB;TTD_MultiTarget
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08253 MMP2 Homo sapiens Human PF00040 PF00045 PF00413 7.7 pIC50 TTD_MultiTarget
Q9ULZ9 MMP17 Homo sapiens Human PF00045 PF00413 PF01471 7.7 pIC50 TTD_MultiTarget
P03956 MMP1 Homo sapiens Human PF00045 PF00413 PF01471 6.1 IC50 ChEMBL;BindingDB