Molecule Details
InChIKeyBLVMGNGXAWHZQW-UHFFFAOYSA-N
Compound Name2-[4-[3-(1H-indol-3-yl)piperidin-1-yl]butyl]-4-phenylpyrido[1,2-c]pyrimidine-1,3-dione
Canonical SMILESO=c1c(-c2ccccc2)c2ccccn2c(=O)n1CCCCN1CCCC(c2c[nH]c3ccccc23)C1
Clinical Status Data-mined Candidate
Targets (Human+Pathogen)3
Pfam Stratification Homologous
Avg pChEMBL6.79
SourceChEMBL;BindingDB
2D Structure
2D structure
Activity Profile
Target Activities (3)
Target Gene Organism Category Pfam pChEMBL Type Source
P08908 HTR1A Homo sapiens Human PF00001 7.7 Ki ChEMBL;BindingDB
P28223 HTR2A Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB
P50406 HTR6 Homo sapiens Human PF00001 6.4 Ki ChEMBL;BindingDB